Pilaralisib (XL147) 95 Well Clear Polystyrene High Bind Stripwell

Pilaralisib (XL147) 95 Well Clear Polystyrene High Bind StripwellPilaralisib (XL147) is a selective and reversible class I PI3K inhibitor for PI3K? ? ? with IC50 of 39 nM 36 nM 23 nM in cell free assays, less potent to PI3K?. Phase 1 2.

Tanespimycin (17-AAG) is a potent HSP90 inhibitor with IC50 of 5 nM in a cell-free assay

also inhibits human P450 isoenzymes CYP2C9

most notably roses

Also inhibiting components of the ubiquitin system

weakly inhibits CYP2A6 and CYP2E1

Milnacipran inhibits both norepinephrine transporter (NET) and norepinephrine transporter (SERT) with IC50 of 77 nM and 420 nM

Felbamate (Felbatol) is an anticonvulsant drug used in the treatment of epilepsy

It is an antimetabolite antineoplastic agent that inhibits the synthesis of DNA

5 nM and 8 nM

Exenatide Acetate

Selinexor (KPT-330) is an orally bioavailable selective CRM1 inhibitor

Corning These 50mL PYREX® graduated cylinders are calibrated "to deliver" (TD) in accordance with ASTM E-1272 and ASTM E-542